{"id":23662,"date":"2025-04-13T17:40:11","date_gmt":"2025-04-13T17:40:11","guid":{"rendered":"https:\/\/researchchemicalstore.eu\/?post_type=product&#038;p=23662"},"modified":"2025-10-22T15:01:37","modified_gmt":"2025-10-22T15:01:37","slug":"flualprasolaami-1-mg-graanulid","status":"publish","type":"product","link":"https:\/\/researchchemicalstore.eu\/et\/product\/flualprasolaami-1-mg-graanulid\/","title":{"rendered":"Flualprasolaam 1 MG graanulid"},"content":{"rendered":"<div id=\"content_tab_description\" class=\"tab-content tab-description\">\n<div class=\"tab-content-inner\">\n<div class=\"tab-content-scroll\">\n<h1><strong>Flualprasolaam 1 MG graanulid \u2013 tugeva bensodiasepiini aktiivsusega uurimisaine<\/strong><\/h1>\n<p><strong>Toote nimi:<\/strong> Flualprasolaam 1 MG graanulid<br \/>\n<strong>Keemiline klass:<\/strong> Triasolobensodiasepiin<br \/>\n<strong>Valem:<\/strong> C17H12ClFN4<br \/>\n<strong>Molekulaarmass:<\/strong> 342,8 g\/mol<br \/>\n<strong>Puhtus:<\/strong> \u2265 98% (HPLC-ga kontrollitud)<br \/>\n<strong>Vorm:<\/strong> 1 mg mikropressitud pelletid<\/p>\n<hr \/>\n<h2><strong>Kirjeldus<\/strong><\/h2>\n<p>Flualprasolaam on tugev bensodiasepiinide klassi kuuluv \u00fchend ja struktuurilt sarnane alprasolaamiga (Xanax), mille eristavaks tunnuseks on fen\u00fc\u00fclts\u00fcklile lisatud fluori aatom. See peen keemiline modifikatsioon suurendab selle afiinsust GABAA retseptorite suhtes, mis suurendab selle tugevust ja pikendab toimeaega.<\/p>\n<p>Flualprasolaam 1 MG pelletid on t\u00e4pselt doseeritud ja m\u00f5eldud ainult <strong>anal\u00fc\u00fctilistel eesm\u00e4rkidel, v\u00f5rdlusuuringuteks ja laborianal\u00fc\u00fcsideks<\/strong>. Ei ole ette n\u00e4htud inimtoiduks.<\/p>\n<hr \/>\n<h2><strong>Rakendused ja uurimist\u00f6\u00f6 eesm\u00e4rgid<\/strong><\/h2>\n<ul>\n<li>GABAergiliste interaktsioonide farmakod\u00fcnaamiline uuring<\/li>\n<li>Retseptori sidumise uuringud ja v\u00f5rdlus teiste triasolobensodiasepiinidega<\/li>\n<li>K\u00e4itumisuuringud loommudelites kontrollitud tingimustes<\/li>\n<li>Stabiilsuse ja lahustuvuse anal\u00fc\u00fcs erinevates lahustites<\/li>\n<li>Referents toksikoloogilistes v\u00f5i anal\u00fc\u00fctilistes laborites (GC-MS\/LC-MS kalibreerimine)<\/li>\n<\/ul>\n<hr \/>\n<h2><strong>Teadlaste eelised<\/strong><\/h2>\n<p>\u2705 <strong>Suur potentsiaal<\/strong> \u2013 Katsekeskkonnas m\u00e4rgatavate efektide saavutamiseks on vaja v\u00e4ikest annust<br \/>\n\u2705 <strong>Stabiilne pelletikuju<\/strong> - Lihtne doseerida ja s\u00e4ilitada<br \/>\n\u2705 <strong>Laboris testitud puhtus<\/strong> \u2013 J\u00e4rjepidevus tagatud reprodutseeritavate uurimistulemuste jaoks<\/p>\n<hr \/>\n<h2><strong>Puudused ja riskid<\/strong><\/h2>\n<p>\u26a0\ufe0f <strong>V\u00e4ga tugev<\/strong> \u2013 Isegi v\u00e4ikesed k\u00f5rvalekalded annuses v\u00f5ivad katsete tulemusi oluliselt m\u00f5jutada<br \/>\n\u26a0\ufe0f <strong>Pikaajaline m\u00f5ju<\/strong> \u2013 V\u00f5ib korduval manustamisel loommudelites akumuleeruda<br \/>\n\u26a0\ufe0f <strong>Vajadus konditsioneeritud ladustamise j\u00e4rele<\/strong> \u2013 Hoida eelistatavalt temperatuuril alla 25 \u00b0C, kuivas ja pimedas.<\/p>\n<hr \/>\n<h2><strong>Kasutus- ja laborijuhised<\/strong><\/h2>\n<ul>\n<li><strong>Soovitatav laboratoorne annus:<\/strong> In vitro testide puhul alustage annusega 0,25\u20130,5 mg. \u00c4rge \u00fcletage seda taset ilma kalibreerimiseta.<\/li>\n<li><strong>Lahustuvus:<\/strong> Lahustub h\u00e4sti etanoolis, DMSO-s ja prop\u00fcleengl\u00fckoolis<\/li>\n<li><strong>S\u00e4ilitamistingimused:<\/strong> Hoida \u00f5hukindlas anumas, jahedas ja otsese p\u00e4ikesevalguse eest kaitstult.<\/li>\n<li><strong>K\u00e4itlemine:<\/strong> Pulbri v\u00f5i lahuse k\u00e4itlemisel kandke kindaid, kaitseprille ja t\u00f6\u00f6tage t\u00f5mbekappi all.<\/li>\n<\/ul>\n<hr \/>\n<h2><strong>Korduma kippuvad k\u00fcsimused (KKK)<\/strong><\/h2>\n<h3>\u2753 <em>Kas flualprasolaam on Hollandis v\u00f5i Belgias legaalne?<\/em><\/h3>\n<p>\u27a1\ufe0f \u00d5iguslik staatus on erinev. Kontrollige alati uusimaid kohalikke eeskirju. \u00dcldiselt on selle tarbimine keelatud, kuid anal\u00fc\u00fctiliseks testimiseks v\u00f5ib see olla lubatud.<\/p>\n<h3>\u2753 <em>Kas ma saan flualprasolaami kasutada une v\u00f5i \u00e4revuse uurimiseks?<\/em><\/h3>\n<p>\u27a1\ufe0f Ainult rangelt kontrollitud laborikeskkonnas ja eranditult mitte-inimmudelitel v\u00f5i keemilise interaktsiooni uuringutes.<\/p>\n<h3>\u2753 <em>Kui kaua p\u00fcsib flualprasolaam toatemperatuuril stabiilsena?<\/em><\/h3>\n<p>\u27a1\ufe0f Kuivas ja pimedas s\u00e4ilib see temperatuuril 20\u201325 \u00b0C v\u00e4hemalt 12 kuud.<\/p>\n<h3>\u2753 <em>Kas esineb ristresistentsust teiste bensodiasepiinidega?<\/em><\/h3>\n<p>\u27a1\ufe0f Jah, flualprasolaamil on kattuvad seondumisprofiilid teiste ainetega, n\u00e4iteks alprasolaami ja klonasolaamiga.<\/p>\n<hr \/>\n<h2><strong>Laboriaruande kokkuv\u00f5te<\/strong><\/h2>\n<table>\n<thead>\n<tr>\n<th>Parameeter<\/th>\n<th>V\u00e4\u00e4rtus<\/th>\n<\/tr>\n<\/thead>\n<tbody>\n<tr>\n<td><strong>Partii number<\/strong><\/td>\n<td>FLPZ-0725<\/td>\n<\/tr>\n<tr>\n<td><strong>Puhtus (HPLC)<\/strong><\/td>\n<td>99,3%<\/td>\n<\/tr>\n<tr>\n<td><strong>V\u00e4limus<\/strong><\/td>\n<td>Valge kristalliline pulber (pressitud graanuliteks)<\/td>\n<\/tr>\n<tr>\n<td><strong>Sulamistemperatuur<\/strong><\/td>\n<td>225\u2013230 \u00b0C<\/td>\n<\/tr>\n<tr>\n<td><strong>Identifitseerimine<\/strong><\/td>\n<td>NMR ja MS abil kinnitatud<\/td>\n<\/tr>\n<\/tbody>\n<\/table>\n<hr \/>\n<h2><strong>Hoiatus<\/strong><\/h2>\n<p><strong>Ei ole ette n\u00e4htud inimtoiduks ega meditsiiniliseks kasutamiseks. Ainult professionaalseks uurimist\u00f6\u00f6ks kvalifitseeritud laborites.<\/strong><\/p>\n<\/div>\n<\/div>\n<\/div>","protected":false},"excerpt":{"rendered":"<h3><span data-sheets-value=\"{\" data-sheets-userformat=\"{\"><span style=\"vertical-align: inherit;\"><span style=\"vertical-align: inherit;\">Flualprazolam Pellets Properties<\/span><\/span><\/span><\/h3>\n<p><strong><span style=\"vertical-align: inherit;\"><span style=\"vertical-align: inherit;\">Synonym:<\/span><\/span><\/strong><span style=\"vertical-align: inherit;\"><span style=\"vertical-align: inherit;\"> Fluclazolam <\/span><\/span><br \/>\n<strong><span style=\"vertical-align: inherit;\"><span style=\"vertical-align: inherit;\">CAS Number:<\/span><\/span><\/strong><span style=\"vertical-align: inherit;\"><span style=\"vertical-align: inherit;\"> 28910-91-0 <\/span><\/span><br \/>\n<strong><span style=\"vertical-align: inherit;\"><span style=\"vertical-align: inherit;\">Formula:<\/span><\/span><\/strong><span style=\"vertical-align: inherit;\"><span style=\"vertical-align: inherit;\"> 8-chloro-6-(2-fluorophenyl)-1-methyl-4H-[1,2,4]triazolo[4,3-a][1,4]benzodiazepine <\/span><\/span><br \/>\n<strong><span style=\"vertical-align: inherit;\"><span style=\"vertical-align: inherit;\">Molar mass:<\/span><\/span><\/strong><span style=\"vertical-align: inherit;\"><span style=\"vertical-align: inherit;\"> 326.8 g\/mol <\/span><\/span><br \/>\n<strong><span style=\"vertical-align: inherit;\"><span style=\"vertical-align: inherit;\">Purity:<\/span><\/span><\/strong><span style=\"vertical-align: inherit;\"><span style=\"vertical-align: inherit;\"> &gt;97%<\/span><\/span><\/p>\n","protected":false},"featured_media":28782,"comment_status":"closed","ping_status":"closed","template":"","meta":[],"product_brand":[],"product_cat":[488],"product_tag":[326],"class_list":["post-23662","product","type-product","status-publish","has-post-thumbnail","product_cat-verboden","product_tag-nl","first","instock","taxable","shipping-taxable","purchasable","product-type-simple"],"_links":{"self":[{"href":"https:\/\/researchchemicalstore.eu\/et\/wp-json\/wp\/v2\/product\/23662","targetHints":{"allow":["GET"]}}],"collection":[{"href":"https:\/\/researchchemicalstore.eu\/et\/wp-json\/wp\/v2\/product"}],"about":[{"href":"https:\/\/researchchemicalstore.eu\/et\/wp-json\/wp\/v2\/types\/product"}],"replies":[{"embeddable":true,"href":"https:\/\/researchchemicalstore.eu\/et\/wp-json\/wp\/v2\/comments?post=23662"}],"version-history":[{"count":4,"href":"https:\/\/researchchemicalstore.eu\/et\/wp-json\/wp\/v2\/product\/23662\/revisions"}],"predecessor-version":[{"id":25752,"href":"https:\/\/researchchemicalstore.eu\/et\/wp-json\/wp\/v2\/product\/23662\/revisions\/25752"}],"wp:featuredmedia":[{"embeddable":true,"href":"https:\/\/researchchemicalstore.eu\/et\/wp-json\/wp\/v2\/media\/28782"}],"wp:attachment":[{"href":"https:\/\/researchchemicalstore.eu\/et\/wp-json\/wp\/v2\/media?parent=23662"}],"wp:term":[{"taxonomy":"product_brand","embeddable":true,"href":"https:\/\/researchchemicalstore.eu\/et\/wp-json\/wp\/v2\/product_brand?post=23662"},{"taxonomy":"product_cat","embeddable":true,"href":"https:\/\/researchchemicalstore.eu\/et\/wp-json\/wp\/v2\/product_cat?post=23662"},{"taxonomy":"product_tag","embeddable":true,"href":"https:\/\/researchchemicalstore.eu\/et\/wp-json\/wp\/v2\/product_tag?post=23662"}],"curies":[{"name":"t\u00f6\u00f6leht","href":"https:\/\/api.w.org\/{rel}","templated":true}]}}