{"id":23404,"date":"2025-04-13T17:39:42","date_gmt":"2025-04-13T17:39:42","guid":{"rendered":"https:\/\/researchchemicalstore.eu\/?post_type=product&#038;p=23404"},"modified":"2025-10-23T00:58:39","modified_gmt":"2025-10-23T00:58:39","slug":"proskalinhydroklorid","status":"publish","type":"product","link":"https:\/\/researchchemicalstore.eu\/is\/vara\/proskalinhydroklorid\/","title":{"rendered":"Proskal\u00ednh\u00fddr\u00f3kl\u00f3r\u00ed\u00f0"},"content":{"rendered":"<h1><strong>Proskal\u00ednh\u00fddr\u00f3kl\u00f3r\u00ed\u00f0 \u2013 fenet\u00fdlam\u00edn aflei\u00f0a fyrir v\u00edsindaranns\u00f3knir<\/strong><\/h1>\n<p><strong>V\u00f6ruheiti:<\/strong> Proskal\u00ednh\u00fddr\u00f3kl\u00f3r\u00ed\u00f0<br \/>\n<strong>Fullt efnaheiti:<\/strong> 4-pr\u00f3pox\u00fd-3,5-d\u00edmetox\u00fdfenet\u00fdlam\u00ednh\u00fddr\u00f3kl\u00f3r\u00ed\u00f0<br \/>\n<strong>Efnaflokkur:<\/strong> Skipt \u00fat fenet\u00fdlam\u00edn<br \/>\n<strong>Sameindaform\u00fala (HCl salt):<\/strong> C13H21NO3 HCl<br \/>\n<strong>M\u00f3lmassi:<\/strong> \u00b1 275,77 g\/m\u00f3l<br \/>\n<strong>\u00datlit:<\/strong> Hv\u00edtt til lj\u00f3sgult kristalla\u00f0 duft<br \/>\n<strong>Hreinleiki:<\/strong> \u2265 98% (HPLC sta\u00f0fest)<br \/>\n<strong>Samheiti:<\/strong> 3,5-d\u00edmetox\u00fd-4-pr\u00f3pox\u00fdfenet\u00fdlam\u00ednh\u00fddr\u00f3kl\u00f3r\u00ed\u00f0<\/p>\n<hr \/>\n<h2>\ud83e\uddea <strong>Hva\u00f0 er Proskal\u00edn HCl?<\/strong><\/h2>\n<p>Proskal\u00edn er <strong>ge\u00f0r\u00e6nt efnasamband<\/strong> sem tilheyrir <strong>fenet\u00fdlam\u00edn fj\u00f6lskylda<\/strong>, skyld meskal\u00edni og eskal\u00edni. \u00dea\u00f0 hefur <strong>pr\u00f3pox\u00fdh\u00f3pur<\/strong> \u00ed sta\u00f0 metox\u00fd- e\u00f0a etox\u00fdh\u00f3ps, sem gefur sameindinni einstaka bindingarvirkni. H\u00fddr\u00f3kl\u00f3r\u00ed\u00f0salti\u00f0 (HCl) er st\u00f6\u00f0ugasta formi\u00f0 og hentar til notkunar \u00e1 ranns\u00f3knarstofum.<\/p>\n<blockquote><p>\u26a0\ufe0f <em>Ekki \u00e6tla\u00f0 til manneldis. Eing\u00f6ngu til ranns\u00f3kna.<\/em><\/p><\/blockquote>\n<hr \/>\n<h2>\ud83d\udd2c <strong>Notkun \u00ed ranns\u00f3knum<\/strong><\/h2>\n<p>Proscaline HCl er rannsaka\u00f0 \u00e1 eftirfarandi svi\u00f0um:<\/p>\n<ul>\n<li><strong>5-HT2A vi\u00f0taka\u00f6rvun<\/strong> og taugalyfjafr\u00e6\u00f0ileg \u00e1hrif<\/li>\n<li><strong>Samanbur\u00f0arbindingartilraunir<\/strong> me\u00f0 \u00f6\u00f0rum fenet\u00fdlam\u00ednum (eins og meskal\u00edni)<\/li>\n<li><strong>SAR ranns\u00f3knir (byggingar-virkni tengsl)<\/strong> innan ge\u00f0lyfja<\/li>\n<li><strong>Greining \u00e1 hugl\u00e6gum \u00e1hrifum<\/strong> \u00ed st\u00fdr\u00f0um ranns\u00f3knarstoful\u00edk\u00f6num<\/li>\n<\/ul>\n<hr \/>\n<h2>\ud83d\udce6 <strong>R\u00e1\u00f0leggingar um notkun og geymslu<\/strong><\/h2>\n<ul>\n<li><strong>Notkun (eing\u00f6ngu in vitro):<\/strong> D\u00e6miger\u00f0ur styrkur fyrir pr\u00f3fanir: 5\u201325 \u00b5M<\/li>\n<li><strong>Leysni:<\/strong> Leysanlegt \u00ed vatni, etan\u00f3li, metan\u00f3li<\/li>\n<li><strong>Geymsluskilyr\u00f0i:<\/strong> Geymi\u00f0 \u00e1 loft\u00fe\u00e9ttum, dimmum og k\u00f6ldum sta\u00f0 (2\u20138\u00b0C)<\/li>\n<li><strong>St\u00f6\u00f0ugleiki:<\/strong> St\u00f6\u00f0ugt \u00ed 24 m\u00e1nu\u00f0i vi\u00f0 bestu a\u00f0st\u00e6\u00f0ur<\/li>\n<li><strong>\u00d6ryggi:<\/strong> Vinni\u00f0 a\u00f0eins me\u00f0 hl\u00edf\u00f0arb\u00fana\u00f0i og vi\u00f0 ranns\u00f3knarstofua\u00f0st\u00e6\u00f0ur<\/li>\n<\/ul>\n<hr \/>\n<h2>\u274c <strong>M\u00f6gulegir \u00f3kostir og \u00e1h\u00e6tta<\/strong><\/h2>\n<ul>\n<li><strong>Sterkt ge\u00f0virkt efni<\/strong> ef um \u00f3viljandi snertingu e\u00f0a misnotkun er a\u00f0 r\u00e6\u00f0a<\/li>\n<li><strong>Takmarka\u00f0ar kl\u00edn\u00edskar ranns\u00f3knir<\/strong> a\u00f0gengilegt \u2013 a\u00f0allega fr\u00e1sagnir af fr\u00e1s\u00f6gnum<\/li>\n<li><strong>L\u00f6glegt gr\u00e1tt sv\u00e6\u00f0i<\/strong> \u00ed nokkrum l\u00f6ndum<\/li>\n<li><strong>Aflei\u00f0ur af fenet\u00fdlam\u00edni<\/strong> getur haft milliverkanir vi\u00f0 m\u00f3n\u00f3am\u00ednkerfi<\/li>\n<li><strong>Ekki hentugt til d\u00fdratilrauna \u00e1n leyfis<\/strong><\/li>\n<\/ul>\n<hr \/>\n<h2>\ud83e\uddfe <strong>Ranns\u00f3knarstofugreining (s\u00fdnislota)<\/strong><\/h2>\n<p><strong>Lotun\u00famer:<\/strong> PRO-HCL-2025-03<br \/>\n<strong>Greiningarmi\u00f0st\u00f6\u00f0:<\/strong> Synaptix ChemTesting, Holland<br \/>\n<strong>Greiningart\u00f3l:<\/strong><\/p>\n<ul>\n<li>HPLC: Hreinleiki 98,4%<\/li>\n<li>NMR: Sta\u00f0festing \u00e1 byggingarbyggingu<\/li>\n<li>FTIR: Sta\u00f0festing virknih\u00f3pa<\/li>\n<li>GC-MS: Au\u00f0kennispr\u00f3fun<\/li>\n<\/ul>\n<p><strong>Dagsetningargreining:<\/strong> 2025-06-01<br \/>\n<strong>Leifar af leysiefnum:<\/strong> Innan \u00f6ruggra ranns\u00f3knarstofugilda<br \/>\n<strong>\u00deungm\u00e1lmar:<\/strong> Ekki greinanlegt<\/p>\n<hr \/>\n<h2>\u2753 <strong>Algengar spurningar \u2013 Algengar spurningar<\/strong><\/h2>\n<h3>\u2753 Hva\u00f0 gerir proskal\u00edn \u00e1 vi\u00f0takastigi?<\/h3>\n<p>\u00dea\u00f0 virkar sem <strong>\u00f6rvandi \u00e1 5-HT2A vi\u00f0taka<\/strong>, svipa\u00f0 og \u00f6nnur ge\u00f0lyf. N\u00e1kv\u00e6mur verkunarh\u00e1ttur er enn til ranns\u00f3knar.<\/p>\n<h3>\u2753 Er Proscaline l\u00f6glegt \u00ed Hollandi e\u00f0a Belg\u00edu?<\/h3>\n<p>Ekki s\u00e9rstaklega skr\u00e1\u00f0 \u00e1 bannlistum, en g\u00e6ti veri\u00f0 banna\u00f0 skv. <strong>hli\u00f0st\u00e6\u00f0 l\u00f6ggj\u00f6f<\/strong>R\u00e1\u00f0f\u00e6r\u00f0u \u00feig alltaf vi\u00f0 l\u00f6gfr\u00e6\u00f0ing.<\/p>\n<h3>\u2753 Hentar \u00feessi vara fyrir pers\u00f3nulegar tilraunir?<\/h3>\n<p><strong>Nei.<\/strong> \u00deessi vara er eing\u00f6ngu til s\u00f6lu <strong>ranns\u00f3knartilgangi \u00ed st\u00fdr\u00f0u ranns\u00f3knarstofuumhverfi<\/strong>Notkun utan \u00feess kassa er <strong>banna\u00f0 og \u00e1h\u00e6ttusamt<\/strong>.<\/p>\n<h3>\u2753 Hvers vegna er h\u00fddr\u00f3kl\u00f3r\u00ed\u00f0formi\u00f0 nota\u00f0?<\/h3>\n<p>Hinn <strong>HCl saltform<\/strong> er st\u00f6\u00f0ugra, leysanlegra \u00ed vatni og au\u00f0veldara a\u00f0 skammta \u00ed n\u00e1kv\u00e6mum ranns\u00f3knarstofuumhverfi en frj\u00e1ls basi.<\/p>\n<hr \/>\n<h2>\u26a0\ufe0f <strong>Fyrirvari<\/strong><\/h2>\n<p>\u00deessi vara er eing\u00f6ngu \u00e6tlu\u00f0 fyrir <strong>l\u00f6gm\u00e6tar ranns\u00f3knir \u00e1 ranns\u00f3knarstofu<\/strong> og kann <strong>ekki \u00e6tla\u00f0 til notkunar fyrir menn e\u00f0a d\u00fdr<\/strong>Sala til e\u00f0a notkun af \u00f3l\u00f6gr\u00e1\u00f0a einstaklingum er stranglega b\u00f6nnu\u00f0. Birgir ber ekki \u00e1byrg\u00f0 \u00e1 neinum misnotkun e\u00f0a \u00f3vi\u00f0eigandi notkun.<\/p>","protected":false},"excerpt":{"rendered":"<h3>Eiginleikar proskal\u00ednh\u00fddr\u00f3kl\u00f3r\u00ed\u00f0s<\/h3>\n<p><strong>Samheiti:<\/strong> 3,5-d\u00edmetox\u00fd-4-pr\u00f3pox\u00fdfenet\u00fdlam\u00ednh\u00fddr\u00f3kl\u00f3r\u00ed\u00f0<br \/>\n<strong>CAS-n\u00famer:<\/strong> 39201-78-0<br \/>\n<strong>Form\u00fala:<\/strong> 2-{3,5-d\u00edmetox\u00fd-4-pr\u00f3p\u00fdlox\u00fdfen\u00fdl}etan-1-am\u00ednh\u00fddr\u00f3kl\u00f3r\u00ed\u00f0<br \/>\n<strong>M\u00f3lmassi:<\/strong> 275,8 g\/m\u00f3l<br \/>\n<strong>Hreinleiki:<\/strong> &gt;97%<\/p>","protected":false},"featured_media":28847,"comment_status":"closed","ping_status":"closed","template":"","meta":[],"product_brand":[],"product_cat":[322,80,536],"product_tag":[326],"class_list":{"0":"post-23404","1":"product","2":"type-product","3":"status-publish","4":"has-post-thumbnail","6":"product_cat-bijna-verboden","7":"product_cat-fenethylamine","8":"product_cat-proscaline","9":"product_tag-nl","11":"first","12":"instock","13":"taxable","14":"shipping-taxable","15":"purchasable","16":"product-type-variable"},"_links":{"self":[{"href":"https:\/\/researchchemicalstore.eu\/is\/wp-json\/wp\/v2\/product\/23404","targetHints":{"allow":["GET"]}}],"collection":[{"href":"https:\/\/researchchemicalstore.eu\/is\/wp-json\/wp\/v2\/product"}],"about":[{"href":"https:\/\/researchchemicalstore.eu\/is\/wp-json\/wp\/v2\/types\/product"}],"replies":[{"embeddable":true,"href":"https:\/\/researchchemicalstore.eu\/is\/wp-json\/wp\/v2\/comments?post=23404"}],"version-history":[{"count":4,"href":"https:\/\/researchchemicalstore.eu\/is\/wp-json\/wp\/v2\/product\/23404\/revisions"}],"predecessor-version":[{"id":26542,"href":"https:\/\/researchchemicalstore.eu\/is\/wp-json\/wp\/v2\/product\/23404\/revisions\/26542"}],"wp:featuredmedia":[{"embeddable":true,"href":"https:\/\/researchchemicalstore.eu\/is\/wp-json\/wp\/v2\/media\/28847"}],"wp:attachment":[{"href":"https:\/\/researchchemicalstore.eu\/is\/wp-json\/wp\/v2\/media?parent=23404"}],"wp:term":[{"taxonomy":"product_brand","embeddable":true,"href":"https:\/\/researchchemicalstore.eu\/is\/wp-json\/wp\/v2\/product_brand?post=23404"},{"taxonomy":"product_cat","embeddable":true,"href":"https:\/\/researchchemicalstore.eu\/is\/wp-json\/wp\/v2\/product_cat?post=23404"},{"taxonomy":"product_tag","embeddable":true,"href":"https:\/\/researchchemicalstore.eu\/is\/wp-json\/wp\/v2\/product_tag?post=23404"}],"curies":[{"name":"wp","href":"https:\/\/api.w.org\/{rel}","templated":true}]}}