{"id":23116,"date":"2025-04-13T17:39:10","date_gmt":"2025-04-13T17:39:10","guid":{"rendered":"https:\/\/researchchemicalstore.eu\/?post_type=product&#038;p=23116"},"modified":"2025-10-23T03:03:52","modified_gmt":"2025-10-23T03:03:52","slug":"pellet-di-etizolam-da-1-mg","status":"publish","type":"product","link":"https:\/\/researchchemicalstore.eu\/it\/prodotto\/pellet-di-etizolam-da-1-mg\/","title":{"rendered":"Pellet di Etizolam da 1 mg"},"content":{"rendered":"<h1><strong><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\">Pellet di Etizolam da 1 MG \u2013 Formulazione di ricerca di grado di laboratorio di tienodiazepine<\/span><\/span><\/strong><\/h1>\n<h2><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\">Panoramica di Etizolam<\/span><\/span><\/h2>\n<p><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\">L&#039;etizolam \u00e8 un analogo delle tienodiazepine con potenti propriet\u00e0 ansiolitiche, sedative e miorilassanti. Questi pellet da 1 mg sono stati sviluppati per studi controllati sulle interazioni con il recettore GABA-A e sui processi neurofarmacologici. <\/span><\/span><a href=\"https:\/\/researchchemicalstore.eu\/it\/negozio\/lisergamidi\/1v-lsd-150-mcg-blotters\/\"><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\">Blotter 1V-LSD 150 MCG<\/span><\/span><\/a><\/p>\n<h2><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\">Caratteristiche del prodotto<\/span><\/span><\/h2>\n<ul>\n<li><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\">Esattamente 1 mg di Etizolam per pellet (variazione \u00b12%)<\/span><\/span><\/li>\n<li><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\">Formulato con cellulosa microcristallina<\/span><\/span><\/li>\n<li><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\">Imballaggi fotostabili e resistenti all&#039;umidit\u00e0<\/span><\/span><\/li>\n<li><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\">Controllo batch per:<\/span><\/span>\n<ul>\n<li><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\">Purezza HPLC (\u226598%)<\/span><\/span><\/li>\n<li><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\">Verifica dell&#039;identit\u00e0 MS<\/span><\/span><\/li>\n<li><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\">Uniformit\u00e0 di peso e dimensioni<\/span><\/span><\/li>\n<\/ul>\n<\/li>\n<\/ul>\n<h2><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\">Profilo farmacologico<\/span><\/span><\/h2>\n<ul>\n<li><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\">Elevata affinit\u00e0 per i recettori GABA-A<\/span><\/span><\/li>\n<li><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\">Legame selettivo ai sottotipi \u03b11\u2013\u03b15<\/span><\/span><\/li>\n<li><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\">Azione farmacologica:<\/span><\/span>\n<ul>\n<li><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\">Ansiolitico<\/span><\/span><\/li>\n<li><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\">Sedativo<\/span><\/span><\/li>\n<li><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\">Rilassante muscolare<\/span><\/span><\/li>\n<\/ul>\n<\/li>\n<li><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\">Emivita di eliminazione pi\u00f9 breve rispetto alle benzodiazepine classiche<\/span><\/span><\/li>\n<\/ul>\n<h2><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\">Aree di applicazione nella ricerca<\/span><\/span><\/h2>\n<ol>\n<li><strong><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\">Neurofarmacologia<\/span><\/span><\/strong>\n<ul>\n<li><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\">Interazioni del recettore GABA-A<\/span><\/span><\/li>\n<li><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\">Modulazione allosterica<\/span><\/span><\/li>\n<li><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\">Specificit\u00e0 del sottotipo<\/span><\/span><\/li>\n<\/ul>\n<\/li>\n<li><strong><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\">Analisi comparativa<\/span><\/span><\/strong>\n<ul>\n<li><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\">Confronto struttura-attivit\u00e0 con le benzodiazepine<\/span><\/span><\/li>\n<li><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\">Ricerca sui percorsi metabolici<\/span><\/span><\/li>\n<\/ul>\n<\/li>\n<li><strong><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\">Scienze comportamentali<\/span><\/span><\/strong>\n<ul>\n<li><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\">Modelli di ansia (ad esempio EPM, OFT)<\/span><\/span><\/li>\n<li><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\">Cicli di sonno e veglia<\/span><\/span><\/li>\n<li><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\">Soppressione delle convulsioni<\/span><\/span><\/li>\n<\/ul>\n<\/li>\n<\/ol>\n<h2><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\">Specifiche tecniche<\/span><\/span><\/h2>\n<ul>\n<li><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\">Diametro del pellet: 2,5 mm \u00b1 0,1 mm<\/span><\/span><\/li>\n<li><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\">Peso: 10 mg \u00b1 0,5 mg<\/span><\/span><\/li>\n<li><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\">Colore: Bianco puro<\/span><\/span><\/li>\n<li><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\">Solubilit\u00e0: &gt;5 mg\/ml in etanolo (96%)<\/span><\/span><\/li>\n<li><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\">Punto di fusione: 146\u2013148\u00b0C<\/span><\/span><\/li>\n<\/ul>\n<h3><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\">Profilo di stabilit\u00e0<\/span><\/span><\/h3>\n<ul>\n<li><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\">Durata di conservazione: 36 mesi a 15\u201325\u00b0C<\/span><\/span><\/li>\n<li><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\">Solidit\u00e0 alla luce: &lt;1% degradazione\/anno<\/span><\/span><\/li>\n<li><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\">Contenuto di umidit\u00e0: &lt;0,5% (Karl Fischer)<\/span><\/span><\/li>\n<\/ul>\n<h2><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\">Linee guida sul dosaggio (solo per riferimento)<\/span><\/span><\/h2>\n<ul>\n<li><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\">In vitro: 10\u20131000 nM<\/span><\/span><\/li>\n<li><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\">Preclinico: 0,05\u20130,5 mg\/kg<\/span><\/span><\/li>\n<li><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\">Modelli comportamentali: 0,1\u20131,0 mg\/kg<\/span><\/span><\/li>\n<\/ul>\n<h2><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\">Informazioni sulla sicurezza e sulla conservazione<\/span><\/span><\/h2>\n<ul>\n<li><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\">Conservare in un imballaggio a prova di luce<\/span><\/span><\/li>\n<li><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\">Umidit\u00e0 relativa &lt;40%<\/span><\/span><\/li>\n<li><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\">Temperatura tra 15\u201325\u00b0C<\/span><\/span><\/li>\n<li><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\">Compatibile con PBS, NaCl 0.9% <\/span><\/span><a href=\"https:\/\/researchchemicalstore.eu\/it\/negozio\/pellet-2\/o-pellet-dsmt-50mg\/\"><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\">Pellet di O-DSMT da 50 mg<\/span><\/span><\/a><\/li>\n<\/ul>\n<h2><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\">Documentazione alla consegna<\/span><\/span><\/h2>\n<ul>\n<li><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\">Certificato di autenticit\u00e0 con:<\/span><\/span>\n<ul>\n<li><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\">Purezza<\/span><\/span><\/li>\n<li><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\">Tempo di conservazione<\/span><\/span><\/li>\n<li><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\">Identificazione di massa<\/span><\/span><\/li>\n<\/ul>\n<\/li>\n<li><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\">Scheda di sicurezza (SDS) secondo GHS<\/span><\/span><\/li>\n<li><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\">Scheda tecnica con:<\/span><\/span>\n<ul>\n<li><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\">Dati di stabilit\u00e0<\/span><\/span><\/li>\n<li><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\">Proposte di progettazione sperimentale<\/span><\/span><\/li>\n<li><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\">Analisi di solubilit\u00e0<\/span><\/span><\/li>\n<\/ul>\n<\/li>\n<\/ul>\n<p><em><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\">Solo per scopi scientifici. Non adatto a scopi medici, diagnostici o al consumo umano. <\/span><\/span><a href=\"https:\/\/researchchemicalstore.eu\/it\/negozio\/top-10-research-chemicals\/caluanie-muelear-ossida\/\"><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\">Caluanie Muelear Ossida<\/span><\/span><\/a><\/em><\/p>","protected":false},"excerpt":{"rendered":"<h2><span style=\"vertical-align: inherit;\"><span style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\">Etizolam pellets properties<\/span><\/span><\/span><\/span><\/h2>\n<p><strong><span style=\"vertical-align: inherit;\"><span style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\">Synonym<\/span><\/span><\/span><\/span><\/strong><span style=\"vertical-align: inherit;\"><span style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\"> : 4-(2-chlorophenyl)-2-ethyl-9-methyl-6H-thieno[3,2-f][1,2,4]triazolo[4,3-a][1,4]diazepine <\/span><\/span><\/span><\/span><br \/>\n<strong><span style=\"vertical-align: inherit;\"><span style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\">CAS Number<\/span><\/span><\/span><\/span><\/strong><span style=\"vertical-align: inherit;\"><span style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\"> : 40054-69-1 <\/span><\/span><\/span><\/span><br \/>\n<strong><span style=\"vertical-align: inherit;\"><span style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\">Formula<\/span><\/span><\/span><\/span><\/strong><span style=\"vertical-align: inherit;\"><span style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\"> : C17H15ClN4S <\/span><\/span><\/span><\/span><br \/>\n<strong><span style=\"vertical-align: inherit;\"><span style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\">Molar mass<\/span><\/span><\/span><\/span><\/strong><span style=\"vertical-align: inherit;\"><span style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\"> : 342.8 g\/mol <\/span><\/span><\/span><\/span><br \/>\n<strong><span style=\"vertical-align: inherit;\"><span style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\">Purity<\/span><\/span><\/span><\/span><\/strong><span style=\"vertical-align: inherit;\"><span style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\"><span dir=\"auto\" style=\"vertical-align: inherit;\"> : \u2265 99%<\/span><\/span><\/span><\/span><\/p>\n","protected":false},"featured_media":28778,"comment_status":"closed","ping_status":"closed","template":"","meta":[],"product_brand":[82],"product_cat":[488],"product_tag":[917,326],"class_list":["post-23116","product","type-product","status-publish","has-post-thumbnail","product_brand-research-chemical","product_cat-verboden","product_tag-etizolam","product_tag-nl","first","instock","taxable","shipping-taxable","purchasable","product-type-simple"],"_links":{"self":[{"href":"https:\/\/researchchemicalstore.eu\/it\/wp-json\/wp\/v2\/product\/23116","targetHints":{"allow":["GET"]}}],"collection":[{"href":"https:\/\/researchchemicalstore.eu\/it\/wp-json\/wp\/v2\/product"}],"about":[{"href":"https:\/\/researchchemicalstore.eu\/it\/wp-json\/wp\/v2\/types\/product"}],"replies":[{"embeddable":true,"href":"https:\/\/researchchemicalstore.eu\/it\/wp-json\/wp\/v2\/comments?post=23116"}],"version-history":[{"count":6,"href":"https:\/\/researchchemicalstore.eu\/it\/wp-json\/wp\/v2\/product\/23116\/revisions"}],"predecessor-version":[{"id":28492,"href":"https:\/\/researchchemicalstore.eu\/it\/wp-json\/wp\/v2\/product\/23116\/revisions\/28492"}],"wp:featuredmedia":[{"embeddable":true,"href":"https:\/\/researchchemicalstore.eu\/it\/wp-json\/wp\/v2\/media\/28778"}],"wp:attachment":[{"href":"https:\/\/researchchemicalstore.eu\/it\/wp-json\/wp\/v2\/media?parent=23116"}],"wp:term":[{"taxonomy":"product_brand","embeddable":true,"href":"https:\/\/researchchemicalstore.eu\/it\/wp-json\/wp\/v2\/product_brand?post=23116"},{"taxonomy":"product_cat","embeddable":true,"href":"https:\/\/researchchemicalstore.eu\/it\/wp-json\/wp\/v2\/product_cat?post=23116"},{"taxonomy":"product_tag","embeddable":true,"href":"https:\/\/researchchemicalstore.eu\/it\/wp-json\/wp\/v2\/product_tag?post=23116"}],"curies":[{"name":"wp","href":"https:\/\/api.w.org\/{rel}","templated":true}]}}